A new synthesis of 2-(aminoalkyl)-1,2,4-triazolo[1,5- a ]pyrimidines

A new synthesis of 2-(aminoalkyl)-1,2,4-triazolo[1,5- a ]pyrimidines Full article

Journal

Mendeleev Communications
ISSN: 1364-551X , E-ISSN: 0959-9436

Output data

Year: 2017, Volume: 27, Number: 2, Pages: 169-171 Pages count : 3 DOI: 10.1016/j.mencom.2017.03.021

Authors

Prezent Mikhail A. ¹ , Daeva Elena D. ¹ , Baranin Sergey V. ¹ , Zavarzin Igor V. ¹

Affiliations

1	N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 119991 Moscow, Russian Federation

Nickel(ii) acetylacetonate-promoted cycloaddition between Boc-protected amino acid hydrazides and benzoylcyanamide followed by deprotection gives 2-amino-5-aminoalkyl-1,2,4-triazoles, whose reaction with 1,3-dielectrophiles affords the title compounds.

Prezent M.A. , Daeva E.D. , Baranin S.V. , Zavarzin I.V.
A new synthesis of 2-(aminoalkyl)-1,2,4-triazolo[1,5- a ]pyrimidines
Mendeleev Communications. 2017. V.27. N2. P.169-171. DOI: 10.1016/j.mencom.2017.03.021 WOS Scopus OpenAlex

≡ Web of science:	WOS:000398749600021
≡ Scopus:	2-s2.0-85016012933
≡ OpenAlex:	W2600299837