Synthesis of 3-acetyl-2-amino-4-pyridone

Synthesis of 3-acetyl-2-amino-4-pyridone Full article

Journal

Russian Chemical Bulletin
ISSN: 1573-9171 , E-ISSN: 1066-5285

Output data

Year: 1996, Volume: 45, Number: 1, Pages: 168-170 Pages count : 3 DOI: 10.1007/bf01433755

Authors

Dorokhov V.A. ¹ , Komkov A.V. ¹ , Sakharov A.M. ¹ , Bogdanov V.S. ¹

Affiliations

1	N. D. Zelinaky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 117913, Moscow, Russian Federation

A method hxsynthesizing 3-acetyl-2-amino-4-pyyridone has been suggested. The synthesis involves the condensation of dimethylformamide dimethylacetal at the NH2 group of diphenylboron chelate diacetylketene aminal followed by its intramolecular cyclization under the action of NaOMe in MeOH.

Dorokhov V.A. , Komkov A.V. , Sakharov A.M. , Bogdanov V.S.
Synthesis of 3-acetyl-2-amino-4-pyridone
Russian Chemical Bulletin. 1996. V.45. N1. P.168-170. DOI: 10.1007/bf01433755 WOS Scopus OpenAlex

≡ Web of science:	WOS:A1996UG35200034
≡ Scopus:	2-s2.0-0042467135
≡ OpenAlex:	W1994161966